|
Vascular Molecular Bioengineering Laboratory The Vascular Bioengineering Laboratory at UCSD Bioengineering was established in 1988 when Dr. Shu Chien and several of his colleagues moved from Columbia University to San Diego. The Laboratory has grown from less than ten staff members to over twenty over the past decade. Our research goal is to elucidate the molecular mechanisms of the regulation of vascular functions, with a special emphasis on the transduction of mechanical stimuli, such as pressure and flow, into intracellular signaling and the ensuing gene expression and functional responses in health and disease. Vascular
endothelial cells (ECs) are continuously exposed to blood flow and
distending pressure, which exert significant influences on physiological
and pathophysiological processes. For instance, the regional variations
in blood flow pattern play a significant role in the preferential
localization of atherosclerosis at arterial branch points. Studies are
conducted at different levels of the biological hierarchy, from
molecules and cells to tissues and animal models, by using a combination
of biological and engineering approaches. Our current emphases are on
the following subjects: Use
of DNA Microarray Technology to Study Gene Expression: Recent
advances in DNA microarray technology provide a powerful and efficient
tool to decipher the complex patterns of gene expression in response to
physical and chemical stimuli by comparing expression levels of
thousands of genes under controlled experimental conditions. We have
investigated the modulation of gene expression in ECs by shear stress
and in smooth muscle cells (SMCs) by matrix geometry. We have
demonstrated that long-term laminar shear stress (24 hr) down-regulates
a number of genes to keep ECs in a relatively quiescent stage. Only a
few genes are up-regulated, mainly those related to EC survival,
angiogenesis and vascular remodeling. These findings provide a better
understanding of the molecular basis of the protection of ECs from
atherogenesis by long-term laminar shear stress, which occurs in the
straight part of the arterial tree. We currently have a dedicated facility that supports all
microarray-related experimentations, with human, rat and mouse cDNA and
oligonucleotide libraries and a platform to perform bioinformatics
analysis. Mechanotransduction
in Endothelial Cells: We are interested in the mechanisms by which
cells sense mechanical stimuli and transduce them into biochemical
signals, especially the mechano-sensor system that initiates the
transduction process. Membrane receptors on both the luminal side (e.g.,
Flk-1), abluminal side (e.g., integrins) of the EC have been found to be
activated by shear stress and play a role in mechanotransduction. Our
results indicate that these receptors interact with each other as a
network to regulate the downstream signaling pathways. Integrins
trans-activate Flk-1 in response to shear stress, but not vice versa.
Integrins also play a role in the control of integrity of intercellular
junction proteins. We studied membrane fluidity on the EC luminal surface as
another potential source of mechano-sensing.
Besides shear stress, we are investigating the mechanism by which
mechanical strain affects molecular and cellular events. We found that
equibiaxial strain with high magnitude (>25%) induced SMC apoptosis
(programmed cell death), whereas lesser strain within physiological
range (<10%) had a protective effect. SMCs subjected to uniaxial
strain aligned in the direction perpendicular to the strain vector, and
the induced JNK expression was transient. In contrast, SMCs subjected to
equibiaxial strain did not undergo any alignment, and the induced JNK
expression was sustained. Thus, uniaxial and equibiaxial strains have
different effects on cell morphologies and cell signaling. We are
currently investigating the molecular mechanisms causing such
differential cellular responses to different modes of mechanical
stimulation. Endothelial
Cell Migration: The migration of vascular cells plays an important
role in many physiological processes. We used a wound-healing model to
investigate the mechanical and molecular mechanisms regulating EC
migration by scraping a strip in an EC monolayer and subsequently
exposing this monolayer to flow. EC strip wounding induced the
dissociation of cell junctions at wound edges. Under laminar flow, more
of the cells upstream to the wound lost their cell junctions, became
dissociated from EC monolayer, and migrated with a great speed into the
wound area along the flow direction, as compared with static cells. The
results suggest that laminar flow promotes EC migration through the
activation of signaling pathways, in addition to a mechanical pushing
effect. In order to dissect
out the various factors, we studied the migration of subconfluent ECs,
which do not have cell-cell adhesions. The migration speed of cells
seeded on different concentrations of extracellular matrix (ECM)
proteins showed a bell-shaped curve, with a peak at an optimal ECM
concentration, indicating that a balance between the attachment at the
cell front and detachment at the cell rear is important for cell
migration. By studying EC migration on ECM proteins seeded on top of an
elastic gel embedded with fluorescently labeled beads, we are mapping
the mechanical strain induced in the membrane and the force exerted by
the migrating cell. The role of Rho small GTPases, which play
significant roles in regulating the cytoskeleton (especially actin
filaments), in cell migration is also being investigated. The dominant
negative mutants of both RhoA and Rac significantly retarded EC
migration and reduced the wound-healing rate. Microtubules, as one of
the components of cytoskeleton, also play an important role in EC
migration, as evidenced by the inhibition of migration with Taxol, a
microtubule-stabilizing agent. In-vivo Investigations: We applied our knowledge from in
vitro studies to in vivo
animal models. We found that a dominant negative mutant of Ras (Ras N17)
blocked the re-stenosis induced by balloon injury of rat arteries,
suggesting a potential role of Ras in gene therapy for the prevention of
re-stenosis after balloon injury. Investigations on signaling pathways in vivo are being conducted in animal models of balloon injury and
hypertension, which is created by banding of the abdominal aorta. The
effects on cellular signaling and gene expression are correlated with
physiological changes. In summary, by using
a systematic approach to study the effects of mechanical stimuli on
mechanosensing, signal transduction, gene expression, cellular dynamics,
and physiological functions, we aim at elucidating the molecular basis
of mechanotransduction in health and disease.
|